SCHEMBL790084

SCHEMBL790084

Nc1nc2ccc(I)cc2c(F)c1-c1ccc(C(=O)N2CCOCC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.48
GRM2 Q14416 1/20 0.46
ATR Q13535 3/20 0.46
KCNH2 Q12809 3/20 0.44
HPGD P15428 4/20 0.44
ERN1 O75460 1/20 0.44
HDAC4 P56524 1/20 0.43
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
PIK3CA P42336 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789847 0.85 JAK2 (0.46) JAK2GRM2ATRKCNH2HPGD
SCHEMBL790716 0.84 MAPT (0.43) HPGDKDM4EALDH1A1SMN1; SMN2
SCHEMBL807223 0.80 IRAK4 (0.46) JAK2ATRKCNH2HPGDPIK3CA
SCHEMBL10277681 0.74 LRRK2 (0.47) JAK2ATRKDM4EALDH1A1SMN1; SMN2
SCHEMBL789402 0.74 CYP1A2 (0.41) HPGDKDM4EALDH1A1CYP1A2
SCHEMBL109082 0.71 PHGDH (0.69) HPGDKDM4EALDH1A1SMN1; SMN2
SCHEMBL807334 0.69 KCNH2 (0.54) JAK2GRM2ATRKCNH2HPGD
SCHEMBL4355847 0.68 JAK2 (0.56) JAK2GRM2KCNH2HPGDERN1
SCHEMBL24547937 0.68 HPGD (0.46) JAK2GRM2HPGDKDM4EALDH1A1
SCHEMBL8172365 0.67 EPHX2 (0.71) HPGDERN1HDAC4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed