SCHEMBL789402

SCHEMBL789402

Nc1nc2ccc(I)cc2c(F)c1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.41
CYP1A1 P04798 2/20 0.41
CYP1B1 Q16678 2/20 0.41
KDM4E B2RXH2 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MAPK1 P28482 2/20 0.41
MAPT P10636 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP2C9 P11712 1/20 0.40
ADORA2A P29274 2/20 0.38
KMT2A Q03164 2/20 0.38
ATM Q13315 1/20 0.38
TLR9 Q9NR96 1/20 0.38
PTGFR P43088 2/20 0.38
DHODH Q02127 1/20 0.37
NPSR1 Q6W5P4 2/20 0.37
HTT P42858 2/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL790716 0.80 MAPT (0.43) KDM4EL3MBTL1MAPK1MAPTTDP1
SCHEMBL790609 0.78 LMNA (0.48) PTGFRDHODH
SCHEMBL790933 0.78 APP (0.47) CYP1A2CYP1A1CYP1B1KDM4EL3MBTL1
SCHEMBL790759 0.78 KDM4E (0.47) KDM4EADORA2ANPSR1HTTHPGD
SCHEMBL789718 0.78 CYP1A1 (0.41) CYP1A2CYP1A1CYP1B1KDM4EL3MBTL1
SCHEMBL790753 0.76 CYP1A2 (0.37) CYP1A2CYP1A1CYP1B1KDM4EL3MBTL1
SCHEMBL28041579 0.73 DHODH (0.49) CYP1A2KDM4EL3MBTL1MAPK1MAPT
SCHEMBL27556561 0.73 CYP1A1 (0.69) CYP1A2CYP1A1CYP1B1MAPTADORA2A
SCHEMBL29058866 0.72 ESR1 (0.64) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL790927 0.71 APP (0.37) MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed