SCHEMBL790716

SCHEMBL790716

Nc1nc2ccc(I)cc2c(F)c1-c1ccc(N2CCOCC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TP53 P04637 1/20 0.43
ALOX15 P16050 1/20 0.43
KDM4E B2RXH2 5/20 0.42
ALDH1A1 P00352 4/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
HPGD P15428 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
AHR P35869 1/20 0.42
MAPK1 P28482 1/20 0.42
GAA P10253 3/20 0.41
HCRTR1 O43613 1/20 0.41
LMNA P02545 1/20 0.41
NCF1 P14598 1/20 0.41
XDH P47989 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL790839 0.83 ADORA2A (0.49) MAPTNPC1RAB9ASMN1; SMN2TP53
SCHEMBL10277681 0.82 LRRK2 (0.47) MAPTNPC1RAB9ASMN1; SMN2TP53
SCHEMBL789402 0.80 CYP1A2 (0.41) MAPTKDM4EALDH1A1L3MBTL1HPGD
SCHEMBL9954672 0.71 TDO2 (0.52) MAPTNPC1RAB9ASMN1; SMN2TP53
SCHEMBL789847 0.69 JAK2 (0.46) SMN1; SMN2KDM4EALDH1A1HPGDADORA2A
SCHEMBL14694267 0.68 ADK (0.41) MAPTNPC1RAB9ASMN1; SMN2TP53
SCHEMBL9954881 0.67 TDO2 (0.52) MAPTNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL1432961 0.67 AKR1C3 (0.65) MAPTNPC1RAB9ASMN1; SMN2TP53
SCHEMBL807328 0.65 KDM4E (0.53) MAPTNPC1RAB9ASMN1; SMN2TP53
SCHEMBL31079126 0.64 MAPT (0.46) MAPTNPC1RAB9ASMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed