SCHEMBL7900939

SCHEMBL7900939

CC(=O)NCCn1c(C2CCCN(C(=O)C[C@@H](Cc3ccc(Br)cc3)NC(=O)OC(C)(C)C)C2)cc2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.37
KDM4E B2RXH2 1/20 0.37
PROKR1 Q8TCW9 5/20 0.37
KLK5 Q9Y337 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ACE P12821 1/20 0.35
CACNA1B Q00975 1/20 0.35
PADI4 Q9UM07 3/20 0.35
CNR2 P34972 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
AKT1 P31749 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2790320 0.90 KDM4E (0.42) TP53KDM4EPROKR1POLBMAPT
SCHEMBL7891183 0.89 PADI4 (0.40) PROKR1KLK5ACECACNA1BPADI4
SCHEMBL7893386 0.89 PROKR1 (0.38) PROKR1KLK5ACECACNA1BPADI4
SCHEMBL762687 0.82 HRH1 (0.41) TP53POLBCTSSCTSKCYP3A4
SCHEMBL2790219 0.80 PADI4 (0.41) PROKR1KLK5ACEPADI4CNR2
SCHEMBL7901541 0.80 PADI4 (0.36) PROKR1KLK5ACEPADI4CNR2
SCHEMBL2817635 0.80 PROKR1 (0.39) TP53PROKR1POLBMAPTSMN1; SMN2
SCHEMBL2791612 0.80 PROKR1 (0.39) TP53PROKR1POLBMAPTSMN1; SMN2
SCHEMBL2790508 0.79 FPR2 (0.34) TP53KDM4ESMN1; SMN2ITGB3ITGA2B
SCHEMBL763469 0.79 HRH1 (0.45) TP53KLK5POLBCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed