SCHEMBL7901870

SCHEMBL7901870

CN(C(=O)N1C=NC(c2cccc(C(=O)NOCc3ccccc3)c2)C1)C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 5/20 0.47
SIGMAR1 Q99720 3/20 0.40
DRD2 P14416 3/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
HTR2B P41595 2/20 0.40
KMT2A Q03164 2/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
MEN1 O00255 1/20 0.39
CCR3 P51677 1/20 0.39
DRD4 P21917 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7894622 0.90 HDAC1 (0.50) KDM1ASIGMAR1DRD2HTR2AHTR2C
SCHEMBL7904409 0.84 SIGMAR1 (0.52) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL7902404 0.83 CCR5 (0.49) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL425436 0.78 KDM1A (0.44) KDM1ASIGMAR1DRD2HTR2AHTR2C
SCHEMBL446158 0.78 DRD2 (0.47) KDM1ASIGMAR1DRD2HTR2AHTR2C
SCHEMBL7901721 0.76 KCNH2 (0.44) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL14938277 0.74 KDM1A (0.49) KDM1ASIGMAR1DRD2HTR2AHTR2C
SCHEMBL14937747 0.70 SLC5A7 (0.42) KDM1ADRD2DRD4NPC1RAB9A
SCHEMBL530727 0.67 FAAH (0.54) KMT2ANPC1RAB9A
SCHEMBL425287 0.66 HDAC1 (0.52) SIGMAR1DRD2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010074588-A2 PHARMACEUTICAL COMPOUNDS BIAL - PORTELA & Cª, S.A. (PT) 2010-07-01 WO disclosed