SCHEMBL7901932

SCHEMBL7901932

COCCCn1c(C2CCCN(C(=O)C[C@@H](Cc3ccc(Br)cc3)NC(=O)OC(C)(C)C)C2)c(C)c2cc(OC)ccc21

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.34
CACNA1B Q00975 2/20 0.33
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33
KLK5 Q9Y337 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7899697 0.91 PROKR1 (0.39) CACNA1BHRH2HRH1KLK5ALDH1A1
SCHEMBL7905913 0.85 CACNA1B (0.35) CACNA1BHRH2HRH1KLK5ALDH1A1
SCHEMBL7891211 0.84 PROKR1 (0.42) HRH2HRH1KLK5ALDH1A1CNR2
SCHEMBL2788383 0.84 KLK5 (0.36) CACNA1BHRH2HRH1KLK5CNR2
SCHEMBL7902566 0.83 PROKR1 (0.38) HRH2HRH1KLK5CNR2
SCHEMBL2789222 0.82 PROKR1 (0.41) ALDH1A1LMNACNR2
SCHEMBL2814433 0.82 PROKR1 (0.39) HRH2HRH1KLK5ALDH1A1CNR2
SCHEMBL2814434 0.82 PROKR1 (0.39) HRH2HRH1KLK5ALDH1A1CNR2
SCHEMBL7896929 0.82 CACNA1B (0.33) CACNA1BHRH2HRH1KLK5ALDH1A1
SCHEMBL7906019 0.81 PDE2A (0.34) CACNA1BHRH2HRH1KLK5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed