SCHEMBL7902076

SCHEMBL7902076

CC1CC2(CCN(C(=O)C3=CC=C(C4=CC=C(F)CC4)CC3)CC2)C(=O)N1[C@@H](C)c1ccc(F)cc1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 6/20 0.34
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
MAPT P10636 1/20 0.30
CCR5 P51681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7907303 0.73 MC4R (0.40)
SCHEMBL7908417 0.60 KIT (0.40) CYP3A4CYP2C9CYP2C19
SCHEMBL4092929 0.55 HSD11B1 (0.49) HSD11B1CYP3A4CYP2C9CYP2C19
SCHEMBL17611772 0.55 OPRM1 (0.38) HSD11B1CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL8023232 0.54 PSEN1 (0.49) HSD11B1CYP3A4CYP2C9CYP2C19
SCHEMBL19416252 0.54 LTA4H (0.44) MAPT
SCHEMBL12685149 0.54 HSD11B1 (0.54) HSD11B1
SCHEMBL3715276 0.54 HSD11B1 (0.54) HSD11B1
SCHEMBL2873080 0.53 HSD11B1 (0.49) HSD11B1CYP3A4CYP2C9CYP2C19
SCHEMBL672150 0.53 ALDH1A1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed