SCHEMBL7904064

SCHEMBL7904064

Cc1c(C2CCCNC2)[nH]c2c(F)cccc12

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.40
HTR2C P28335 3/20 0.40
KCNH2 Q12809 3/20 0.40
DRD2 P14416 2/20 0.39
DRD3 P35462 1/20 0.38
CCNT1 O60563 4/20 0.38
CDK9 P50750 4/20 0.38
CCNK O75909 2/20 0.37
CCNE1 P24864 2/20 0.37
CDK2 P24941 2/20 0.37
CDK12 Q9NYV4 2/20 0.37
CDK7 P50613 1/20 0.37
CCNH P51946 1/20 0.37
MNAT1 P51948 1/20 0.37
HTR6 P50406 1/20 0.36
HTR1A P08908 1/20 0.36
SLC6A2 P23975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2789459 0.84 CCNT1 (0.41) HTR2AHTR2CKCNH2DRD2DRD3
SCHEMBL7898453 0.78 HTR2A (0.57) HTR2AHTR2CKCNH2DRD2DRD3
SCHEMBL16760180 0.78 HTR2A (0.57) HTR2AHTR2CKCNH2DRD2DRD3
SCHEMBL2791447 0.74 CYP2D6 (0.41) HTR2AHTR2CKCNH2CCNT1CDK9
SCHEMBL7901873 0.70 CCNT1 (0.45) HTR2AHTR2CKCNH2DRD2DRD3
SCHEMBL7901095 0.69 HPGDS (0.46) HTR6
SCHEMBL2789373 0.68 HTR2A (0.42) HTR2AHTR2CKCNH2DRD2CCNT1
SCHEMBL2788485 0.68 CCNT1 (0.51) HTR2AHTR2CKCNH2DRD2DRD3
SCHEMBL2145272 0.67 HTR6 (0.45) HTR2ADRD2DRD3HTR6HTR1A
SCHEMBL7897980 0.67 HTR6 (0.46) HTR2AHTR2CHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed