SCHEMBL790545

SCHEMBL790545

COc1ncc(-c2ccc3nc(N)c(C(=O)N4CCC5(CC4)OCCO5)cc3c2)cc1S(=O)(=O)NCC1CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 3/20 0.44
POLB P06746 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 7/20 0.43
CYP3A4 P08684 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP2C19 P33261 1/20 0.43
PI4KA P42356 3/20 0.41
PIK3CG P48736 3/20 0.41
KDM4E B2RXH2 1/20 0.40
RAB9A P51151 1/20 0.39
PIK3R1 P27986 1/20 0.39
PIK3CA P42336 1/20 0.39
TP53 P04637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
GAA P10253 2/20 0.35
HPGD P15428 1/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL791568 0.90 PI4KA (0.43) PIK3C3POLBALDH1A1CYP3A4CYP2C19
SCHEMBL12474809 0.89 PI4KA (0.41) PIK3C3POLBALDH1A1CYP3A4CYP2C19
SCHEMBL807161 0.88 PIK3C3 (0.49) PIK3C3POLBALDH1A1PI4KAPIK3CG
SCHEMBL806791 0.88 PI4KA (0.43) PIK3C3POLBALDH1A1CYP3A4CYP2C19
SCHEMBL789808 0.85 PIK3CG (0.44) PIK3C3POLBALDH1A1PI4KAPIK3CG
SCHEMBL807111 0.85 RAB9A (0.46) POLBKMT2AALDH1A1PI4KAPIK3CG
SCHEMBL807023 0.85 PIK3CG (0.49) PIK3C3PI4KAPIK3CGRAB9APIK3R1
SCHEMBL789820 0.84 ALDH1A1 (0.43) PIK3C3POLBALDH1A1CYP3A4CYP2C19
SCHEMBL789741 0.84 PI4KA (0.46) POLBALDH1A1PI4KAPIK3CGKDM4E
SCHEMBL807010 0.84 SMN1; SMN2 (0.44) PIK3C3POLBALDH1A1PI4KAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed