SCHEMBL7905583

SCHEMBL7905583

COC(=O)[C@H](C)NC(=O)c1cc(C(F)(F)F)cc(N)c1N

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CFTR P13569 2/20 0.45
CTSS P25774 2/20 0.40
CTSK P43235 2/20 0.40
ALDH1A1 P00352 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
BCL2L1 Q07817 1/20 0.38
P2RX1 P51575 1/20 0.36
SCN9A Q15858 3/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MAPK1 P28482 1/20 0.35
EGLN1 Q9GZT9 2/20 0.35
CNR2 P34972 2/20 0.35
CNR1 P21554 1/20 0.35
ALOX5AP P20292 2/20 0.35
FEN1 P39748 2/20 0.35
LNPEP Q9UIQ6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9310483 0.86 EGLN1 (0.46) CFTRCTSSCTSKALDH1A1NPSR1
SCHEMBL9310492 0.86 EGLN1 (0.46) CFTRCTSSCTSKALDH1A1NPSR1
SCHEMBL7904464 0.84 ALDH1A1 (0.49) ALDH1A1P2RX1HPGDMAPK1
SCHEMBL31113950 0.77 NPSR1 (0.54) NPSR1BCL2L1P2RX1MAPK1
SCHEMBL27883930 0.77 CFTR (0.67) CFTRALDH1A1P2RX1KDM4EHPGD
SCHEMBL5102312 0.73 MLYCD (0.53) NPSR1
SCHEMBL9311399 0.73 ALDH1A1 (0.50) ALDH1A1P2RX1KDM4EHPGDMAPK1
SCHEMBL9311405 0.73 ALDH1A1 (0.50) ALDH1A1P2RX1KDM4EHPGDMAPK1
SCHEMBL31160842 0.71 KEAP1 (0.49) ALDH1A1BCL2L1SCN9AKDM4EHPGD
SCHEMBL18106794 0.71 MAOA (0.41) ALDH1A1BCL2L1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6201119-B1 2,3,4,5-TETRAHYDRO-1H-1,4-BENZODIAZEPIN-9-AMINE COMPOUNDS USEFUL AS INTERMEDIATES TO ANTIVIRALS JANSSEN PHARMACEUTICA N.V. (BE) 2001-03-13 US disclosed