SCHEMBL7907928

SCHEMBL7907928

N=C(N)N1CCN(C(=O)NCC(=O)Nc2cccc(C(=O)NCCC(=O)O)c2)CC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.45
ITGB3 P05106 6/20 0.43
ITGA2B P08514 5/20 0.43
NAMPT P43490 1/20 0.43
ITGA2 P17301 1/20 0.42
EPHX2 P34913 2/20 0.42
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TMPRSS2 O15393 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TPSAB1 Q15661 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SMYD3 Q9H7B4 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8385319 0.91 NAMPT (0.47) NAMPTEPHX2HTTL3MBTL1TMPRSS2
SCHEMBL7909721 0.91 POLB (0.46) GAAITGB3ITGA2BNAMPTITGA2
SCHEMBL7913448 0.90 GAA (0.45) GAANAMPTEPHX2KMT2ASMYD3
SCHEMBL7900164 0.87 MEN1 (0.50) GAAITGB3ITGA2BITGA2EPHX2
SCHEMBL8386581 0.87 FAAH (0.44) HTTL3MBTL1TMPRSS2SMN1; SMN2MEN1
SCHEMBL7909446 0.86 SMN1; SMN2 (0.49) GAAITGB3ITGA2BITGA2EPHX2
SCHEMBL7900157 0.86 ITGB3 (0.51) GAAITGB3ITGA2BNAMPTITGA2
SCHEMBL8381689 0.85 EPHX2 (0.53) ITGB3ITGA2BNAMPTEPHX2HTT
SCHEMBL8386238 0.84 HTT (0.43) NAMPTEPHX2HTTL3MBTL1SMN1; SMN2
SCHEMBL9337540 0.84 GAA (0.53) GAAITGB3ITGA2BITGA2EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608759-B1 Piperazine derivatives MERCK PATENT GMBH (DE) 2001-08-22 EP disclosed
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed
EP-0608759-A2 Piperazinderivatives MERCK PATENT GmbH (DE) 1994-08-03 EP disclosed