SCHEMBL7908500

SCHEMBL7908500

Nc1nc(N2CCOCC2)nn1-c1nnc(-c2ccccc2O)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.41
MAPT P10636 1/20 0.39
AR P10275 1/20 0.38
MTOR P42345 4/20 0.37
PIK3CG P48736 2/20 0.37
PIK3CD O00329 1/20 0.37
PKM P14618 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PTPN11 Q06124 2/20 0.35
TRPM8 Q7Z2W7 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
PIK3R1 P27986 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tetrabuthylammonium SCHEMBL7908484 0.89 TSHR (0.36) PIK3CAMAPTARMTORPIK3CG
SCHEMBL7902640 0.89 NR1I2 (0.43) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL7896551 0.80 CNR2 (0.36) PIK3CAMAPTARMTORPIK3CD
SCHEMBL7908481 0.78 PIK3CB (0.44) PIK3CAMAPTMTORPIK3CDKDM4E
SCHEMBL7904007 0.75 USP2 (0.40) KDM4EALDH1A1SMN1; SMN2
SCHEMBL7896426 0.74 MAPK1 (0.42) ALDH1A1GAAPTPN11TRPM8NPC1
SCHEMBL7905773 0.72 BACE1 (0.39) KDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL1207814 0.71 AR (0.58) MAPTARGAAPTPN11NPC1
SCHEMBL7902631 0.70 RAB9A (0.38) MAPTGLAGAAHPGDHSD17B10
SCHEMBL7896508 0.70 HRH3 (0.41) MAPTKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191152-B1 CARDIOVASCULAR DISORDERS, NERVOUS SYSTEM DISORDERS EGIS GYÓGYSZERGYAR RT. (HU) 2001-02-20 US disclosed
EP-0958294-A1 2-(1,2,4-TRIAZOLE-1-YL)-1,3,4-THIADIAZOLE DERIVATIVES HAVING AN EFFECT ON THE C.N.S. AND THE HEART EGIS GYOGYSZERGYAR (HU) 1999-11-24 EP disclosed
WO-1998030561-A1 2-(1,2,4-TRIAZOLE-1-YL)-1,3,4-THIADIAZOLE DERIVATIVES HAVING AN EFFECT ON THE C.N.S. AND THE HEART EGIS Gyógyszergyár Rt. (HU) 1998-07-16 WO disclosed