SCHEMBL79094

SCHEMBL79094

CCC(CC)CSc1ccccc1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.42
P4HB P07237 1/20 0.41
BACE1 P56817 1/20 0.39
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
EPHX2 P34913 1/20 0.36
LMNA P02545 4/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
HSD17B10 Q99714 2/20 0.35
POLB P06746 2/20 0.33
ALOX15 P16050 2/20 0.33
CA2 P00918 2/20 0.33
CA4 P22748 2/20 0.33
NPC1 O15118 1/20 0.33
CA12 O43570 1/20 0.33
GMNN O75496 1/20 0.33
EGFR P00533 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78524 0.83 TSHR (0.46) TSHRP4HBBACE1MAOAMAOB
SCHEMBL20067971 0.80 P4HB (0.46) TSHRP4HBBACE1MAOAMAOB
SCHEMBL11855729 0.78 P4HB (0.45) TSHRP4HBBACE1MAOAMAOB
SCHEMBL1128730 0.77 P4HB (0.42) TSHRP4HBEPHX2LMNAKDM4E
SCHEMBL6068906 0.76 P4HB (0.43) TSHRP4HBBACE1MAOAMAOB
SCHEMBL6068909 0.76 P4HB (0.43) TSHRP4HBBACE1MAOAMAOB
SCHEMBL10504004 0.74 PTGS2 (0.51) TSHRP4HBEPHX2LMNAKDM4E
SCHEMBL8397211 0.72 LMNA (0.45) TSHRP4HBBACE1EPHX2LMNA
SCHEMBL68951 0.72 HSPA5 (0.46) TSHRP4HBBACE1EPHX2LMNA
SCHEMBL12610426 0.71 MAOA (0.57) MAOAMAOBLMNAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8618162-B2 Insecticidal carbamates exhibiting species-selective inhibition of acetylcholinesterase (AChE) VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. (US) 2013-12-31 US disclosed
US-20120122970-A1 INSECTICIDAL CARBAMATES EXHIBITING SPECIES-SELECTIVE INHIBITION OF ACETYLCHOLINESTERASE (AChE) VIRGINIA POLYTECHNIC INSTITUTE AND STATE UNIVERSITY 2012-05-17 US disclosed
US-8129428-B2 Insecticidal carbamates exhibiting species-selective inhibition of acetylcholinesterase (AChE) VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. (US) 2012-03-06 US disclosed
WO-2009036235-A2 INSECTICIDAL CARBAMATES EXHIBITING SPECIES-SELECTIVE INHIBITION OF ACETYLCHOLINESTERASE (ACHE) VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. (US) 2009-03-19 WO disclosed
US-20090068242-A1 INSECTICIDAL CARBAMATES EXHIBITING SPECIES-SELECTIVE INHIBITION OF ACETYLCHOLINESTERASE (AChE) VIRGINIA POLYTECHNIC INSTITUTE AND STATE UNIVERSITY 2009-03-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090068242-A1 INSECTICIDAL CARBAMATES EXHIBITING SPECIES-SELECTIVE INHIBITION OF ACETYLCHOLINESTERASE (AChE) ACHE, BCHE, CHAT TSHR 1442/4885P4HB 3656/4885BACE1 121/4885
US-20120122970-A1 INSECTICIDAL CARBAMATES EXHIBITING SPECIES-SELECTIVE INHIBITION OF ACETYLCHOLINESTERASE (AChE) ACHE, BCHE, CHAT TSHR 1442/4885P4HB 3656/4885BACE1 121/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.