SCHEMBL7912394

SCHEMBL7912394

COc1ccc(C(=O)CC(NC(=O)C(F)(F)F)C(=O)O)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 6/20 0.47
TAS1R1 Q7RTX1 6/20 0.47
LMNA P02545 2/20 0.43
ATM Q13315 1/20 0.43
ALDH1A1 P00352 2/20 0.42
KMT2A Q03164 2/20 0.42
RECQL P46063 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
KCNH2 Q12809 1/20 0.41
KMO O15229 1/20 0.40
PRSS1 P07477 1/20 0.40
TMPRSS15 P98073 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7899441 1.00 TAS1R3 (0.47) TAS1R3TAS1R1LMNAATMALDH1A1
SCHEMBL7821304 0.90 CYP1A2 (0.48) LMNAATMALDH1A1KMT2ASMN1; SMN2
SCHEMBL7821313 0.90 CYP1A2 (0.48) LMNAATMALDH1A1KMT2ASMN1; SMN2
SCHEMBL5351455 0.87 HTT (0.50) TAS1R3TAS1R1LMNAALDH1A1KMT2A
SCHEMBL5889370 0.87 HTT (0.50) TAS1R3TAS1R1LMNAALDH1A1KMT2A
SCHEMBL5355623 0.87 HTT (0.50) TAS1R3TAS1R1LMNAALDH1A1KMT2A
SCHEMBL7899412 0.86 KMO (0.56) LMNAALDH1A1HTTKMO
SCHEMBL7907206 0.86 KMO (0.56) LMNAALDH1A1HTTKMO
SCHEMBL7907182 0.86 KMO (0.56) LMNAALDH1A1HTTKMO
SCHEMBL7905593 0.80 KMO (0.46) TAS1R3TAS1R1SMN1; SMN2KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207709-B1 FOR THERAPY AND PROPHYLAXIS OF NEURODEGENERATIVE DISEASES, SUCH AS HUNTINGTON'S CHOREA, ALZHEIMER'S DISEASE, DEMENTIA CAUSED BY AQUIRED IMMUNODEFICIENCY SYNDROME (AIDS), INFARCTUAL DEMENTIA, CEREBRAL ISCHEMIA, CEREBRAL HYPOXIA, EPILEPSY PHARMACIA & UPJOHN S.P.A. (IT) 2001-03-27 US disclosed