SCHEMBL7905593

SCHEMBL7905593

COC(=O)[C@@H](CC(=O)c1ccc(Cl)c(Cl)c1)NC(=O)C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMO O15229 4/20 0.46
TAS1R3 Q7RTX0 2/20 0.42
TAS1R1 Q7RTX1 2/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MCHR1 Q99705 1/20 0.42
HPGD P15428 1/20 0.41
GRN P28799 1/20 0.41
SORT1 Q99523 1/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7907206 0.86 KMO (0.56) KMOSLC6A4SLC6A3GRNSORT1
SCHEMBL7907182 0.86 KMO (0.56) KMOSLC6A4SLC6A3GRNSORT1
SCHEMBL7899412 0.86 KMO (0.56) KMOSLC6A4SLC6A3GRNSORT1
SCHEMBL7912394 0.80 TAS1R3 (0.47) KMOTAS1R3TAS1R1SMN1; SMN2
SCHEMBL7899441 0.80 TAS1R3 (0.47) KMOTAS1R3TAS1R1SMN1; SMN2
SCHEMBL7905591 0.78 KMO (0.48) KMOTAS1R3TAS1R1SLC6A4SLC6A3
SCHEMBL19660202 0.77 KMO (0.56) KMOSLC6A4SLC6A3HPGD
SCHEMBL7405864 0.76 KMO (0.68) KMOSLC6A4SLC6A3HPGD
SCHEMBL7868632 0.76 KMO (0.68) KMOSLC6A4SLC6A3HPGD
SCHEMBL7799556 0.75 ALDH1A1 (0.48) TAS1R3TAS1R1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207709-B1 FOR THERAPY AND PROPHYLAXIS OF NEURODEGENERATIVE DISEASES, SUCH AS HUNTINGTON'S CHOREA, ALZHEIMER'S DISEASE, DEMENTIA CAUSED BY AQUIRED IMMUNODEFICIENCY SYNDROME (AIDS), INFARCTUAL DEMENTIA, CEREBRAL ISCHEMIA, CEREBRAL HYPOXIA, EPILEPSY PHARMACIA & UPJOHN S.P.A. (IT) 2001-03-27 US disclosed