SCHEMBL7913442

SCHEMBL7913442

O=C(O)CCN1CCN(C(=O)CNC(=O)N2CCNCC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.43
ITGA2B P08514 3/20 0.43
KDM1A O60341 2/20 0.38
KMT2A Q03164 2/20 0.38
GLA P06280 1/20 0.37
HTR1A P08908 1/20 0.37
HTR7 P34969 1/20 0.37
TPSAB1 Q15661 1/20 0.36
TPSD1 Q9BZJ3 1/20 0.36
TPSG1 Q9NRR2 1/20 0.36
POLB P06746 1/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
FAAH O00519 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
ALOX12 P18054 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8386948 0.86 KMT2A (0.40) KMT2ATPSAB1TPSD1TPSG1POLB
SCHEMBL7913360 0.82 TPSAB1 (0.37) ITGB3ITGA2BKMT2AGLAHTR1A
SCHEMBL16574883 0.81 ITGB3 (0.48) ITGB3ITGA2BKDM1AGLAHTR1A
SCHEMBL8473161 0.79 CA2 (0.50) KMT2ATPSAB1TPSD1TPSG1POLB
SCHEMBL7528972 0.77 GLA (0.53) ITGB3ITGA2BKMT2AGLAPOLB
Aziridine SCHEMBL28507214 0.76 GLA (0.57) ITGB3ITGA2BKDM1AGLAHTR1A
SCHEMBL16574879 0.75 ITGB3 (0.44) ITGB3ITGA2BKMT2AGLAHTR1A
SCHEMBL7344790 0.75 GLA (0.55) ITGB3ITGA2BKMT2AGLAPOLB
SCHEMBL905223 0.75 GLA (0.55) ITGB3ITGA2BKMT2AGLAPOLB
SCHEMBL13387648 0.73 TPSAB1 (0.42) KMT2ATPSAB1TPSD1TPSG1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608759-B1 Piperazine derivatives MERCK PATENT GMBH (DE) 2001-08-22 EP disclosed
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed
EP-0608759-A2 Piperazinderivatives MERCK PATENT GmbH (DE) 1994-08-03 EP disclosed