SCHEMBL7913360

SCHEMBL7913360

N=C(N)N1CCN(C(=O)NCC(=O)N2CCN(CCC(=O)O)CC2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 2/20 0.37
TPSD1 Q9BZJ3 2/20 0.37
TPSG1 Q9NRR2 2/20 0.37
KMT2A Q03164 2/20 0.37
GLA P06280 1/20 0.36
HTR1A P08908 1/20 0.36
HTR7 P34969 1/20 0.36
ITGB3 P05106 4/20 0.36
ITGA2B P08514 3/20 0.36
MAPK1 P28482 2/20 0.35
KDM4E B2RXH2 1/20 0.35
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
SIGMAR1 Q99720 2/20 0.34
FAAH O00519 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
ALOX12 P18054 1/20 0.34
MTOR P42345 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8386026 0.86 ITGB3 (0.40) TPSAB1TPSD1TPSG1KMT2AITGB3
SCHEMBL7909740 0.86 SMN1; SMN2 (0.46) TPSAB1TPSD1TPSG1KMT2AGLA
SCHEMBL7913442 0.82 ITGB3 (0.43) TPSAB1TPSD1TPSG1KMT2AGLA
SCHEMBL8384455 0.81 PKM (0.45) TPSAB1TPSD1TPSG1GLAHTR1A
SCHEMBL8382720 0.79 KMT2A (0.48) TPSAB1TPSD1TPSG1KMT2AITGB3
SCHEMBL8381872 0.77 PKM (0.40) TPSAB1TPSD1TPSG1KMT2AITGB3
SCHEMBL8384378 0.73 MAPK1 (0.47) HTR1AHTR7ITGB3ITGA2BMAPK1
SCHEMBL18596470 0.71 TDP1 (0.56) KMT2AMAPK1KDM4EDRD2DRD3
SCHEMBL657440 0.70 POLB (0.59) KMT2AGLAHTR1AHTR7ITGB3
SCHEMBL7909434 0.69 SMN1; SMN2 (0.50) TPSAB1TPSD1TPSG1KMT2AGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608759-B1 Piperazine derivatives MERCK PATENT GMBH (DE) 2001-08-22 EP disclosed
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed
EP-0608759-A2 Piperazinderivatives MERCK PATENT GmbH (DE) 1994-08-03 EP disclosed