SCHEMBL7915568

SCHEMBL7915568

CC(C)c1ccc(CN2CCN(C(c3cccc(Cl)c3)c3cccc(Cl)c3)CC2)c(=O)c(NCCO)c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 4/20 0.42
CACNA1B Q00975 4/20 0.42
CACNB1 Q02641 4/20 0.42
CACNA1C Q13936 3/20 0.42
CACNA1G O43497 2/20 0.40
POLB P06746 2/20 0.40
MAPT P10636 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
DRD2 P14416 3/20 0.40
DRD3 P35462 3/20 0.40
CYP3A4 P08684 2/20 0.40
CHRM2 P08172 2/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2C P18825 2/20 0.40
DRD4 P21917 2/20 0.40
HRH2 P25021 2/20 0.40
HTR2A P28223 2/20 0.40
ADRA1A P35348 2/20 0.40
HRH1 P35367 2/20 0.40
OPRK1 P41145 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7921443 0.91 ATM (0.45) DRD2DRD3CYP3A4CHRM2ADRA2A
Hydrochloric Acid SCHEMBL7921978 0.90 MEN1 (0.44) CYP3A4KCNH2USP2CYP1A2CYP2D6
SCHEMBL195024 0.86 LMNA (0.48) CACNA1BPOLBMAPTDRD2DRD3
Hydrochloric Acid SCHEMBL7921655 0.85 LMNA (0.48) CACNA1BPOLBMAPTDRD2DRD3
SCHEMBL7921250 0.84 CACNA1B (0.42) CACNA2D1CACNA1BCACNB1CACNA1CCACNA1G
SCHEMBL7924056 0.82 DRD2 (0.43) CACNA1BMAPTDRD2DRD3CHRM2
SCHEMBL7923980 0.81 SMN1; SMN2 (0.38) MAPTNPSR1DRD2DRD4CYP2D6
SCHEMBL7921833 0.80 TACR1 (0.38) POLBMAPTCYP3A4KCNH2USP2
SCHEMBL7924018 0.80 ALDH1A1 (0.58) MAPTNPSR1MEN1ALOX15KMT2A
SCHEMBL7921879 0.79 MEN1 (0.41) POLBDRD2DRD3CYP3A4CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6221868-B1 Remedies/preventives for frequent urination/urinary incontinence and tropone derivatives NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2001-04-24 US disclosed