SCHEMBL7916997

SCHEMBL7916997

CCOC(=O)N(C(=O)OCC)c1ccc(CC2=CN3C=C(C)NC3C(c3cccc(Cl)c3)=C2)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
DYRK3 O43781 1/20 0.35
DYRK1A Q13627 1/20 0.35
DYRK2 Q92630 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
MAPT P10636 2/20 0.35
GRIN2B Q13224 2/20 0.33
GRIN1 Q05586 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
KCNH2 Q12809 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 2/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7929296 0.84 DYRK3 (0.49) JAK2JAK3DYRK3DYRK1ADYRK2
SCHEMBL7902852 0.83 NPC1 (0.34) DYRK3DYRK1ADYRK2DYRK1BMAPT
SCHEMBL7912990 0.82 PARP1 (0.37) JAK2JAK3DYRK3DYRK1ADYRK2
SCHEMBL7914652 0.81 DYRK3 (0.37) DYRK3DYRK1ADYRK2DYRK1BKMT2A
SCHEMBL7902988 0.81 GRIN1 (0.32) GRIN2BGRIN1SMN1; SMN2NPC1RAB9A
SCHEMBL7915334 0.81 DHFR (0.32) SMN1; SMN2NPC1RAB9A
SCHEMBL7913078 0.80 DYRK3 (0.37) DYRK3DYRK1ADYRK2DYRK1B
SCHEMBL7917981 0.80 DYRK3 (0.35) DYRK3DYRK1ADYRK2DYRK1BGRIN2B
SCHEMBL7902845 0.80 PIM1 (0.31)
SCHEMBL7913253 0.76 MAOB (0.34) MAPTSMN1; SMN2ALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed