SCHEMBL7918923

SCHEMBL7918923

CCOC(=O)C(Oc1c(OC)cc(Br)cc1[N+](=O)[O-])C(=O)OCC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.44
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
TDP1 Q9NUW8 2/20 0.40
KDM4E B2RXH2 2/20 0.40
HTT P42858 1/20 0.39
LMNA P02545 1/20 0.39
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
GAA P10253 2/20 0.38
MAPT P10636 2/20 0.38
MAPK1 P28482 2/20 0.38
TNF P01375 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ABCB1 P08183 1/20 0.37
ABCC1 P33527 1/20 0.37
POLB P06746 1/20 0.37
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7918929 0.81 HTT (0.37) ALDH1A1CYP2C19CYP1A2TDP1HTT
SCHEMBL383187 0.79 L3MBTL1 (0.44) ALDH1A1TDP1KDM4EHTTLMNA
SCHEMBL2088203 0.78 TUBB4A (0.49) ALDH1A1TDP1KDM4EHTTMEN1
SCHEMBL27561415 0.75 CYP3A4 (0.41) ALDH1A1CYP2C19CYP1A2TDP1KDM4E
SCHEMBL3353885 0.74 ALDH1A1 (0.47) ALDH1A1TDP1KDM4EHTTLMNA
SCHEMBL4293853 0.73 ALDH1A1 (0.48) ALDH1A1CYP2C19CYP1A2HTTLMNA
Acetic Acid Methyl Ester SCHEMBL27561416 0.73 LMNA (0.46) ALDH1A1CYP2C19CYP1A2LMNAMEN1
SCHEMBL6975821 0.72 MAPT (0.52) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL7372393 0.72 KMT2A (0.46) ALDH1A1TDP1KDM4EHTTLMNA
SCHEMBL29830329 0.72 MAOB (0.45) ALDH1A1CYP2C19CYP1A2TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6221863-B1 TREATING DEPRESSION IN A PATIENT AMERICAN HOME PRODUCTS CORP. 2001-04-24 US disclosed
WO-2000040581-A1 3,4-DIHYDRO-2H-BENZO[1,4]OXAZINE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-07-13 WO disclosed