SCHEMBL7928447

SCHEMBL7928447

CCCSc1ccc(OB(Oc2ccc(SCCC)cc2)Oc2ccc(SCCC)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA13 Q8N1Q1 1/20 0.46
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
AR P10275 2/20 0.39
ALDH1A1 P00352 6/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 3/20 0.35
MAPK1 P28482 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 1/20 0.35
SLC2A1 P11166 1/20 0.34
DRD2 P14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7922025 0.89 MAOA (0.47) CA12CA1CA2CA7CA13
SCHEMBL7934090 0.87 MAOA (0.42) MAOAMAOBMTNR1AMTNR1BAR
SCHEMBL7928525 0.85 THRB (0.44) MAOAMAOBARMAPTSLC2A1
SCHEMBL7931588 0.85 RAB9A (0.38) CA12CA1CA2CA7CA13
SCHEMBL7928451 0.85 CA12 (0.43) CA12CA1CA2CA7CA13
SCHEMBL5206052 0.83 SLC6A4 (0.41) MAOAMAOBMTNR1AMTNR1BALDH1A1
SCHEMBL13397915 0.81 CA12 (0.50) CA12CA1CA2CA7CA13
SCHEMBL13397872 0.80 CA12 (0.61) CA12CA1CA2CA7CA13
SCHEMBL6123648 0.79 ALDH1A1 (0.54) CA12CA1CA2CA7CA13
SCHEMBL7922029 0.74 MAOA (0.45) MAOAMAOBMTNR1AMTNR1BAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed