SCHEMBL7929587

SCHEMBL7929587

CCOCCN(C)c1ccc(Br)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
GAA P10253 1/20 0.40
TAAR1 Q96RJ0 1/20 0.37
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
CHRM2 P08172 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
CHRM1 P11229 1/20 0.35
DRD1 P21728 1/20 0.35
TBXA2R P21731 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
OPRM1 P35372 1/20 0.35
DRD3 P35462 1/20 0.35
SLC6A3 Q01959 1/20 0.35
ALOX15 P16050 1/20 0.35
THRA P10827 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7929581 0.87 MEN1 (0.38) HPGDTAAR1ALDH1A1KDM4ECHRM2
SCHEMBL27512370 0.81 TAAR1 (0.39) HPGDNPC1RAB9ATAAR1ALDH1A1
SCHEMBL1637985 0.81 ALOX15 (0.43) TAAR1ALDH1A1ALOX15
SCHEMBL6344902 0.78 THRA (0.37) HPGDALDH1A1KDM4EALOX15THRA
SCHEMBL1432529 0.78 TAAR1 (0.43) TAAR1ALDH1A1KDM4ESLC6A2MAPT
SCHEMBL6344900 0.77 ALOX15 (0.35) HPGDALDH1A1KDM4EALOX15THRA
SCHEMBL12086382 0.77 ALOX15 (0.33) ALDH1A1KDM4EALOX15THRAMAPT
SCHEMBL19982794 0.77 ADRA2A (0.37) ADRA2AALOX15THRAMMP14MAPT
SCHEMBL9187621 0.76 S100B (0.49) GAAALDH1A1KDM4EALOX15THRA
SCHEMBL19882559 0.75 KMT2A (0.33) NPC1RAB9AKDM4EALOX15MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed