SCHEMBL7930028

SCHEMBL7930028

Clc1cc(C(Cl)(Cl)Cl)cc(C(Cl)(Cl)Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.44
CYP3A4 P08684 3/20 0.36
MAPK1 P28482 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 2/20 0.35
TP53 P04637 1/20 0.33
HIF1A Q16665 1/20 0.32
RECQL P46063 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7096749 0.93 TSHR (0.53) TSHRCYP3A4MAPK1TDP1ALDH1A1
SCHEMBL7928488 0.91 TSHR (0.50) TSHRCYP3A4MAPK1TDP1ALDH1A1
SCHEMBL1538847 0.86 TSHR (0.47) TSHRCYP3A4MAPK1TDP1
SCHEMBL7928485 0.83 TSHR (0.44) TSHRCYP3A4MAPK1TDP1
SCHEMBL10974819 0.77 TSHR (0.33) TSHRMAPK1TDP1TP53HIF1A
SCHEMBL11611118 0.75 TSHR (0.39) TSHRCYP3A4ALDH1A1TP53
SCHEMBL196785 0.71 TSHR (0.50) TSHRCYP3A4MAPK1TDP1ALDH1A1
SCHEMBL3786224 0.71 RAPGEF4 (0.47) TSHRCYP3A4TDP1ALDH1A1HIF1A
SCHEMBL10183607 0.71 GABRA1 (0.52) TSHRTDP1ALDH1A1HSD17B10
SCHEMBL4113569 0.71 TSHR (0.55) TSHRCYP3A4MAPK1TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6201152-B1 HEATING MIXTURE OF METHYL-3,5-DICHLORO-4-METHYLBENZOATE AND ALPHA,ALPHA,ALPHA-TRICHLOROMETHYLBENZENE IN PRESENCE OF AMMONIUM MOLYBDATE CATALYST OCCIDENTAL CHEMICAL CORPORATION 2001-03-13 US claimed
US-4080378-A REACTING A CARBOXYLIC ACID ESTER WITH A TRICHLOROMETHYL SUBSTITUTED AROMATIC COMPOUND IN THE PRESENCE OF A MOLYBDENUM CATALYST DYNAMIT NOBEL AKTIENGESELLSCHAFT (DT) 1978-03-21 US claimed
US-4079090-A Preparation of trichloromethyl-trifluoro methyl-benzenes BAYER AKTIENGESELLSCHAFT (DT) 1978-03-14 US claimed
US-4163753-A FROM AN ALIPHATIC ACID ANHYDRIDE AND A TRICHLOROMETHYL AROMATIC COMPOUND Diaz Chemical Corporation (US) 1979-08-07 US disclosed
US-4104300-A MOLYBDENUM CATALYST, COMPLEXING AGENT DYNAMIT NOBEL AKTIENGESELLSCHAFT (DE) 1978-08-01 US disclosed
US-4080378-A REACTING A CARBOXYLIC ACID ESTER WITH A TRICHLOROMETHYL SUBSTITUTED AROMATIC COMPOUND IN THE PRESENCE OF A MOLYBDENUM CATALYST DYNAMIT NOBEL AKTIENGESELLSCHAFT (DT) 1978-03-21 US disclosed
US-4079090-A Preparation of trichloromethyl-trifluoro methyl-benzenes BAYER AKTIENGESELLSCHAFT (DT) 1978-03-14 US disclosed