SCHEMBL7930529

SCHEMBL7930529

CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)[N+]1(S(=O)(=O)c2ccccc2)CC2(CCNCC2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 14/20 0.46
OPRM1 P35372 1/20 0.46
ACE P12821 1/20 0.44
TACR2 P21452 4/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
TACR1 P25103 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7654721 0.85 GHSR (0.49) GHSROPRM1ACE
SCHEMBL8462876 0.84 GHSR (0.39) GHSROPRM1ACE
Hydrochloric Acid SCHEMBL7575092 0.83 GHSR (0.42) GHSROPRM1ACETACR1
SCHEMBL7848280 0.78 GHSR (0.37) GHSROPRM1ACE
Hydrochloric Acid SCHEMBL7571696 0.76 GHSR (0.37) GHSRACETACR1
SCHEMBL8161727 0.75 GHSR (0.39) GHSRTACR2TACR1
SCHEMBL7979239 0.74 GHSR (0.39) GHSRACETACR1
SCHEMBL8466975 0.74 GHSR (0.39) GHSRMMP2MMP9TACR1
SCHEMBL9391064 0.74 GHSR (0.50) GHSROPRM1ACE
SCHEMBL7401537 0.74 GHSR (0.45) GHSROPRM1ACEMMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1011667-A4 ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE MERCK & CO INC (US) 2001-03-28 EP disclosed
US-6150352-A ARYLQUINOLONE ANALOGS MERCK & CO., INC. (US) 2000-11-21 US disclosed
EP-1011667-A1 ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE Merck & Co., Inc. (a New Jersey corp.) (US) 2000-06-28 EP disclosed
WO-1998055119-A1 ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE MERCK & CO., INC. (US) 1998-12-10 WO disclosed