SCHEMBL7934151

SCHEMBL7934151

CCOCCOc1ccc(Br)cc1F

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
NSD2 O96028 1/20 0.42
NSD3 Q9BZ95 1/20 0.42
HPGD P15428 2/20 0.42
TSHR P16473 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
GAA P10253 1/20 0.41
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
PKM P14618 1/20 0.40
LMNA P02545 1/20 0.40
AAK1 Q2M2I8 2/20 0.39
NCF1 P14598 1/20 0.38
SLC6A4 P31645 1/20 0.38
KDM1A O60341 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16362049 0.86 SMN1; SMN2 (0.44) ALDH1A1NSD2NSD3HPGDTSHR
SCHEMBL7929556 0.84 ALDH1A1 (0.48) ALDH1A1HPGDTSHRL3MBTL1GAA
SCHEMBL5881114 0.84 HPGD (0.55) ALDH1A1NSD2NSD3HPGDTSHR
SCHEMBL1509935 0.84 HPGD (0.51) ALDH1A1HPGDTSHRL3MBTL1GAA
SCHEMBL29929937 0.83 NSD2 (0.44) NSD2NSD3HPGDL3MBTL1KDM4E
SCHEMBL9340707 0.83 L3MBTL1 (0.46) ALDH1A1HPGDL3MBTL1POLBLMNA
SCHEMBL1311491 0.83 SMN1; SMN2 (0.49) NSD2NSD3HPGDTSHRL3MBTL1
SCHEMBL1823347 0.83 NSD2 (0.44) NSD2NSD3HPGDL3MBTL1KDM4E
SCHEMBL27082290 0.83 ALDH1A1 (0.48) ALDH1A1HPGDTSHRL3MBTL1SMN1; SMN2
SCHEMBL6687682 0.81 SMN1; SMN2 (0.50) NSD2NSD3HPGDL3MBTL1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed