SCHEMBL7934175

SCHEMBL7934175

O=C(O)C1=Cc2cc(-c3ccc(C(F)(F)F)cc3)ccc2S(=O)(=O)CC1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.43
CA9 Q16790 3/20 0.40
CA12 O43570 2/20 0.40
P2RY14 Q15391 4/20 0.38
SLC6A2 P23975 1/20 0.38
CTSL P07711 1/20 0.38
DHODH Q02127 1/20 0.38
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
RXRG P48443 1/20 0.37
GALR1 P47211 1/20 0.36
KIF11 P52732 3/20 0.35
PPARA Q07869 1/20 0.35
LMNA P02545 1/20 0.35
HDAC2 Q92769 1/20 0.34
ACLY P53396 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7931169 0.88 CA12 (0.39) PTGDR2CA9CA12DHODHRXRA
SCHEMBL7974920 0.87 BCL2L1 (0.39) PTGDR2CA9CA12GALR1LMNA
SCHEMBL7969661 0.86 PTGDR2 (0.41) PTGDR2CA9CA12P2RY14CTSL
SCHEMBL7929538 0.85 CA12 (0.43) PTGDR2CA9CA12CTSLDHODH
SCHEMBL7929501 0.84 MCL1 (0.39) PTGDR2CA9CA12DHODHRXRA
SCHEMBL3499284 0.84 ALAD (0.35) PTGDR2CA12RXRARXRBGALR1
SCHEMBL7970423 0.81 HAO1 (0.35) DHODH
SCHEMBL7931034 0.81 MAPT (0.41) CA9CA12DHODHRXRA
SCHEMBL7929550 0.81 RXRA (0.37) DHODHRXRARXRBRXRGKIF11
SCHEMBL7972312 0.81 CCR5 (0.38) PTGDR2CA9CA12CTSLRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed