SCHEMBL793437

SCHEMBL793437

FC(F)(F)c1ccc2c(c1)CN(c1cnccc1C1CC1)CC2

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 14/20 0.50
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
CCR2 P41597 1/20 0.38
KDM4C Q9H3R0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL793875 0.82 TRPV3 (0.41) HTR2AHTR2C
SCHEMBL794272 0.78 PHGDH (0.43) HTR2AHTR2C
SCHEMBL798567 0.77 CYP17A1 (0.44) CYP17A1
SCHEMBL793796 0.77 CYP17A1 (0.58) CYP17A1
SCHEMBL20776824 0.70 MAPT (0.46)
SCHEMBL798794 0.68 HRH3 (0.40) HTR2AHTR2C
SCHEMBL12065737 0.68 TRPV3 (0.39) CCR2
SCHEMBL13735785 0.67 CYP17A1 (1.00) CYP17A1
SCHEMBL13737172 0.67 CYP17A1 (1.00) CYP17A1
SCHEMBL10078849 0.66 MAOA (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627648-A1 17aHYDROXYLASE/C17,20-LYASE INHIBITORS Novartis AG (CH) 2013-08-21 EP disclosed
WO-2012035078-A1 17α-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2012-03-22 WO disclosed