SCHEMBL793875

SCHEMBL793875

Cc1ccncc1N1CCc2ccc(C(F)(F)F)cc2C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV3 Q8NET8 1/20 0.41
KDR P35968 4/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
NOTUM Q6P988 1/20 0.40
PDGFRB P09619 3/20 0.39
PHGDH O43175 1/20 0.39
JAK2 O60674 2/20 0.38
SRC P12931 2/20 0.38
PDE10A Q9Y233 1/20 0.38
SPR P35270 1/20 0.38
DDR1 Q08345 1/20 0.37
DDR2 Q16832 1/20 0.37
SCN9A Q15858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL794272 0.95 PHGDH (0.43) TRPV3KDRHTR2AHTR2CNOTUM
SCHEMBL798794 0.84 HRH3 (0.40) KDRHTR2AHTR2CJAK2SRC
SCHEMBL793437 0.82 CYP17A1 (0.50) HTR2AHTR2C
SCHEMBL798654 0.81 PDGFRB (0.43) KDRPDGFRB
SCHEMBL793143 0.81 GRIN2D (0.42) KDRPDGFRB
SCHEMBL798533 0.79 TIPARP (0.46) KDRPDGFRBSCN9A
SCHEMBL793474 0.76 CYP11B2 (0.41) KDRHTR2AHTR2CPDGFRBPDE10A
SCHEMBL793461 0.75 CYP11B2 (0.43) HTR2AHTR2CNOTUMJAK2SRC
SCHEMBL12065737 0.75 TRPV3 (0.39) TRPV3KDRNOTUMPHGDHSPR
SCHEMBL793449 0.75 PARP1 (0.42) HTR2AHTR2CNOTUMJAK2SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627648-A1 17aHYDROXYLASE/C17,20-LYASE INHIBITORS Novartis AG (CH) 2013-08-21 EP claimed
WO-2012035078-A1 17α-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2012-03-22 WO claimed