SCHEMBL794272

SCHEMBL794272

Cc1ccncc1N1CCc2cc(C(F)(F)F)ccc2C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 1/20 0.43
KDR P35968 4/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
SCN9A Q15858 1/20 0.40
S1PR1 P21453 1/20 0.40
NOTUM Q6P988 1/20 0.40
JAK2 O60674 2/20 0.38
SRC P12931 2/20 0.38
PDE10A Q9Y233 1/20 0.38
NAMPT P43490 2/20 0.38
PDGFRB P09619 3/20 0.37
TRPV3 Q8NET8 1/20 0.37
ASIC3 Q9UHC3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL793875 0.95 TRPV3 (0.41) PHGDHKDRHTR2AHTR2CSCN9A
SCHEMBL798794 0.79 HRH3 (0.40) KDRHTR2AHTR2CSCN9AS1PR1
SCHEMBL793437 0.78 CYP17A1 (0.50) HTR2AHTR2C
SCHEMBL798654 0.76 PDGFRB (0.43) KDRPDGFRB
SCHEMBL793143 0.76 GRIN2D (0.42) KDRPDGFRB
SCHEMBL793474 0.76 CYP11B2 (0.41) KDRHTR2AHTR2CPDE10APDGFRB
SCHEMBL793461 0.75 CYP11B2 (0.43) HTR2AHTR2CNOTUMJAK2SRC
SCHEMBL793449 0.75 PARP1 (0.42) HTR2AHTR2CNOTUMJAK2SRC
SCHEMBL798533 0.74 TIPARP (0.46) KDRSCN9AS1PR1PDGFRB
SCHEMBL27889387 0.73 PHGDH (0.43) PHGDHKDRSCN9AS1PR1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627648-A1 17aHYDROXYLASE/C17,20-LYASE INHIBITORS Novartis AG (CH) 2013-08-21 EP claimed
WO-2012035078-A1 17α-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2012-03-22 WO claimed