SCHEMBL798654

SCHEMBL798654

Cc1ccncc1N1CCc2ccc(O)cc2C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 3/20 0.43
KDR P35968 3/20 0.43
DRD2 P14416 6/20 0.40
DRD1 P21728 6/20 0.40
DRD5 P21918 5/20 0.40
DRD3 P35462 5/20 0.40
DRD4 P21917 3/20 0.40
ESR1 P03372 2/20 0.39
ESR2 Q92731 2/20 0.39
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
EED O75530 1/20 0.38
GRIN2D O15399 2/20 0.37
GRIN3B O60391 2/20 0.37
GRIN1 Q05586 2/20 0.37
GRIN2A Q12879 2/20 0.37
GRIN2B Q13224 2/20 0.37
GRIN2C Q14957 2/20 0.37
GRIN3A Q8TCU5 2/20 0.37
CHRM1 P11229 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL793143 0.84 GRIN2D (0.42) PDGFRBKDRCYP11B1CYP11B2EED
SCHEMBL798146 0.84 DRD1 (0.42) PDGFRBKDRDRD2DRD1DRD5
SCHEMBL798533 0.82 TIPARP (0.46) PDGFRBKDRDRD2DRD1DRD5
SCHEMBL793875 0.81 TRPV3 (0.41) PDGFRBKDR
SCHEMBL793474 0.79 CYP11B2 (0.41) PDGFRBKDRCYP11B1CYP11B2
SCHEMBL793623 0.77 MAPT (0.52)
SCHEMBL794272 0.76 PHGDH (0.43) PDGFRBKDR
SCHEMBL5518917 0.75 DRD1 (0.50) DRD2DRD1DRD5DRD3DRD4
SCHEMBL793106 0.73 CYP11B2 (0.48) ESR1ESR2CYP11B1CYP11B2
SCHEMBL793768 0.73 CYP11B2 (0.41) ESR1ESR2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627648-A1 17aHYDROXYLASE/C17,20-LYASE INHIBITORS Novartis AG (CH) 2013-08-21 EP disclosed
WO-2012035078-A1 17α-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2012-03-22 WO disclosed