SCHEMBL7939463

SCHEMBL7939463

Cc1ccc(Cc2ncc(CNCCCCC3CCN(Cc4ccccc4)C3=O)[nH]2)c(C#N)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.38
FNTA P49354 11/20 0.34
FNTB P49356 11/20 0.34
PGGT1B P53609 9/20 0.34
ACHE P22303 3/20 0.33
HTR3A P46098 2/20 0.33
CHRNA7 P36544 1/20 0.33
BCHE P06276 2/20 0.33
HTR6 P50406 2/20 0.32
PKM P14618 2/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
ADRB2 P07550 1/20 0.32
CHRM2 P08172 1/20 0.32
ADRB1 P08588 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.32
CHRM1 P11229 1/20 0.32
DRD2 P14416 1/20 0.32
ADRA2B P18089 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7936033 0.86 KCNH2 (0.48) KCNH2FNTAFNTBPGGT1BCYP3A4
SCHEMBL7927442 0.83 FNTA (0.46) KCNH2FNTAFNTBPGGT1BCYP3A4
SCHEMBL7936646 0.69 FNTA (0.52) KCNH2FNTAFNTBPGGT1BPKM
SCHEMBL7937509 0.68 FNTA (0.69) KCNH2FNTAFNTBPGGT1BCYP3A4
Hydrochloric Acid SCHEMBL7939633 0.67 FNTA (0.68) KCNH2FNTAFNTBPGGT1BCYP3A4
Hydrochloric Acid SCHEMBL7939637 0.67 FNTA (0.68) KCNH2FNTAFNTBPGGT1BCYP3A4
SCHEMBL7937336 0.67 FNTA (0.56) KCNH2FNTAFNTBPGGT1B
SCHEMBL7464954 0.65 FNTA (0.45) KCNH2FNTAFNTBPGGT1B
SCHEMBL8965454 0.64 SLC6A2 (0.45) PKMALDH1A1GAA
SCHEMBL8298317 0.63 BRS3 (0.48) BCHEDRD2DRD4OPRM1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001017992-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed