SCHEMBL7945192

SCHEMBL7945192

CCCOc1ccc(C(=O)Nc2cnc3c(c2)CN(C)CC3)cc1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.42
BRAF P15056 11/20 0.42
RAF1 P04049 3/20 0.42
TAAR1 Q96RJ0 1/20 0.42
ROCK2 O75116 1/20 0.41
CYP3A4 P08684 1/20 0.41
WNT3A P56704 1/20 0.41
KIT P10721 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8130753 0.99 HTR2A (0.42) HTR2ABRAFRAF1TAAR1ROCK2
SCHEMBL7945155 0.89 BRAF (0.51) BRAFRAF1ROCK2CYP3A4KIT
SCHEMBL7955614 0.88 BRAF (0.44) HTR2ABRAFRAF1ROCK2SMN1; SMN2
SCHEMBL6295104 0.88 ROCK2 (0.53) HTR2ATAAR1ROCK2CYP3A4KDM4E
SCHEMBL7951743 0.87 MAPT (0.52) HTR2AROCK2CYP3A4SMN1; SMN2KDM4E
SCHEMBL7945228 0.87 ABL1 (0.48) BRAFKIT
SCHEMBL7953997 0.85 ALDH1A1 (0.43) ROCK2CYP3A4KDM4EMAPT
SCHEMBL7953516 0.84 SMN1; SMN2 (0.44) BRAFTAAR1ROCK2WNT3AKIT
SCHEMBL7951869 0.82 EGFR (0.44) BRAFTAAR1ROCK2WNT3ASMN1; SMN2
SCHEMBL7951760 0.79 MAPT (0.61) ROCK2CYP3A4SMN1; SMN2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6245778-B1 1,6-naphthyridine anti-convulsants SMITHKLINE BEECHAM P.L.C. (GB) 2001-06-12 US claimed
US-6245778-B1 1,6-naphthyridine anti-convulsants SMITHKLINE BEECHAM P.L.C. (GB) 2001-06-12 US disclosed
EP-0986559-A1 1,6-NAPHTHYRIDINE ANTI-CONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2000-03-22 EP disclosed
WO-1998054184-A1 1,6-NAPHTHYRIDINE ANTI-CONVULSANTS SMITHKLINE BEECHAM PLC (GB) 1998-12-03 WO disclosed