SCHEMBL7951869

SCHEMBL7951869

CC(C)c1ccc(C(=O)Nc2cnc3c(c2)CN(C)CC3)cc1C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.44
BRAF P15056 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
WNT3A P56704 1/20 0.41
RET P07949 1/20 0.41
ABL1 P00519 4/20 0.41
DDR1 Q08345 3/20 0.41
DDR2 Q16832 3/20 0.41
KDR P35968 2/20 0.41
HSP90AA1 P07900 1/20 0.41
BCR P11274 1/20 0.40
KCNQ3 O43525 1/20 0.40
KCNQ2 O43526 1/20 0.40
KCNE1 P15382 1/20 0.40
KCNQ1 P51787 1/20 0.40
STK10 O94804 1/20 0.40
NTRK1 P04629 1/20 0.40
LCK P06239 1/20 0.40
EPHA2 P29317 1/20 0.40
EPHA8 P29322 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7958472 0.90 ROCK2 (0.42) EGFRBRAFDDR1NTRK1ROCK2
SCHEMBL7955614 0.87 BRAF (0.44) BRAFSMN1; SMN2KCNQ3KCNQ2ROCK2
SCHEMBL7953516 0.87 SMN1; SMN2 (0.44) EGFRBRAFSMN1; SMN2WNT3AABL1
SCHEMBL7945228 0.86 ABL1 (0.48) EGFRBRAFABL1BCR
SCHEMBL7953309 0.86 MAPT (0.42) SMN1; SMN2KDRHSP90AA1ROCK2MAPT
SCHEMBL7945155 0.85 BRAF (0.51) BRAFROCK2
Hydrochloric Acid SCHEMBL6295059 0.85 ROCK2 (0.51) EGFRBRAFROCK2
SCHEMBL7958661 0.82 KDR (0.47) SMN1; SMN2KDRROCK2MAPT
SCHEMBL7945192 0.82 HTR2A (0.42) BRAFSMN1; SMN2WNT3AROCK2TAAR1
Hydrochloric Acid SCHEMBL8130753 0.81 HTR2A (0.42) BRAFSMN1; SMN2WNT3AROCK2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6245778-B1 1,6-naphthyridine anti-convulsants SMITHKLINE BEECHAM P.L.C. (GB) 2001-06-12 US claimed
US-6245778-B1 1,6-naphthyridine anti-convulsants SMITHKLINE BEECHAM P.L.C. (GB) 2001-06-12 US disclosed
EP-0986559-A1 1,6-NAPHTHYRIDINE ANTI-CONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2000-03-22 EP disclosed
WO-1998054184-A1 1,6-NAPHTHYRIDINE ANTI-CONVULSANTS SMITHKLINE BEECHAM PLC (GB) 1998-12-03 WO disclosed