SCHEMBL7946053

SCHEMBL7946053

Cc1cccc(CCn2c3ccc[c]c3c3c(C(N)=O)cccc32)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.39
NR3C2 P08235 1/20 0.38
ADRA1D P25100 1/20 0.38
MAPT P10636 2/20 0.38
MAPK8 P45983 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
ALDH1A1 P00352 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
GAA P10253 1/20 0.36
TP53 P04637 2/20 0.36
TLR8 Q9NR97 1/20 0.36
PARP1 P09874 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
DAO P14920 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7050803 0.91 ADRA1D (0.44) ADRA1DMAPTMAPK8MEN1KMT2A
SCHEMBL7616815 0.88 SIRT2 (0.38) SIRT2NR3C2ADRA1DMAPTMAPK8
SCHEMBL7467933 0.85 RPS6KB1 (0.36) ADRA1DMAPK8MEN1KMT2AALDH1A1
SCHEMBL27508047 0.82 P2RX4 (0.42) MAPTMEN1KMT2AALDH1A1GAA
SCHEMBL7944531 0.82 GPR52 (0.42) DAO
SCHEMBL27506801 0.81 ICMT (0.38) ADRA1DMEN1KMT2AALDH1A1GAA
SCHEMBL27506423 0.80 ADRA1D (0.43) ADRA1DMAPTMAPK8MEN1KMT2A
SCHEMBL7420567 0.80 MEN1 (0.44) ADRA1DMAPTMEN1KMT2AALDH1A1
SCHEMBL6612458 0.80 PLA2G2A (0.44) ADRA1DPARP1
SCHEMBL27507605 0.80 PLA2G2A (0.39) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001066111-A1 COMPOSITIONS CONTAINING POTENTIAL SPLA2 INHIBITORS FOR THE TREATMENT OF PAIN ELI LILLY AND COMPANY (US) 2001-09-13 WO disclosed