SCHEMBL7947101

SCHEMBL7947101

FC(F)(F)c1c(-c2ccccc2)cc(N2CCNCC2)nc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.52
CSNK1D P48730 2/20 0.47
MAPK11 Q15759 2/20 0.47
MAPK14 Q16539 2/20 0.47
CYP1A2 P05177 3/20 0.44
CYP2C19 P33261 1/20 0.44
CYP2C9 P11712 1/20 0.44
HTR6 P50406 3/20 0.43
HTR1A P08908 1/20 0.43
HTR2A P28223 1/20 0.43
HTR7 P34969 1/20 0.43
HTR5A P47898 1/20 0.43
ADRB1 P08588 2/20 0.43
NCF1 P14598 1/20 0.43
ALDH1A1 P00352 2/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1686083 0.82 MET (0.45) ALDH1A1NPSR1KDM4ELMNA
SCHEMBL1686076 0.82 CSNK1D (0.47) ADRB2CSNK1DMAPK11MAPK14CYP1A2
SCHEMBL1686127 0.82 ACVR1 (0.45) ADRB2CSNK1DMAPK11MAPK14CYP1A2
SCHEMBL7943088 0.78 ADRB2 (0.55) ADRB2CYP1A2CYP2C19CYP2C9HTR1A
SCHEMBL1686085 0.76 CKS1B (0.55)
SCHEMBL2954143 0.75 MAPK14 (0.60) ADRB2CSNK1DMAPK11MAPK14CYP1A2
Hydrochloric Acid SCHEMBL2955401 0.74 MAPK14 (0.58) ADRB2CSNK1DMAPK11MAPK14CYP1A2
SCHEMBL10465983 0.73 ADRB1 (0.68) ADRB2CSNK1DMAPK11MAPK14CYP1A2
SCHEMBL10630930 0.73 ADRB1 (0.60) ADRB2CSNK1DMAPK11MAPK14CYP1A2
SCHEMBL27687352 0.73 HTR1A (0.54) ADRB2HTR6HTR1AHTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010012758-A1 PIPERAZIN-1-YL-TRIFLUOROMETHYL-SUBSTITUTED-PYRIDINES AS FAST DISSOCIATING DOPAMINE 2 RECEPTOR ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2010-02-04 WO disclosed