SCHEMBL7951244

SCHEMBL7951244

COC(=O)C(C)(C)CCC(=O)c1ccc(F)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.43
CHRNG P07510 1/20 0.43
CHRNB1 P11230 1/20 0.43
CHRNB2 P17787 1/20 0.43
SLC6A2 P23975 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CHRND Q07001 1/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
ALDH1A1 P00352 4/20 0.41
L3MBTL1 Q9Y468 1/20 0.38
DPP4 P27487 1/20 0.38
RAB9A P51151 4/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3286504 0.85 ALDH1A1 (0.49) ALDH1A1L3MBTL1RAB9AMAPTMEN1
SCHEMBL977134 0.81 SLC6A3 (0.40) SLC6A3CES2CES1ALDH1A1L3MBTL1
SCHEMBL3333245 0.79 ALDH1A1 (0.44) ALDH1A1L3MBTL1RAB9AMAPTHPGD
SCHEMBL15189645 0.77 CES2 (0.48) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL1274789 0.77 NPSR1 (0.50) CES2ALDH1A1RAB9AMEN1KMT2A
SCHEMBL28403586 0.76 CES2 (0.41) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL22039571 0.76 AAK1 (0.40) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL6809579 0.75 CES2 (0.46) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL25193546 0.73 MEN1 (0.54) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL2575501 0.73 CHRNA1 (0.38) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326372-B1 BENIGN PROSTATE HYPERPLASIA MERCK & CO., INC. 2001-12-04 US disclosed