SCHEMBL795359

SCHEMBL795359

CC(=O)NC(C)CC(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
MTNR1A P48039 6/20 0.44
MTNR1B P49286 6/20 0.44
MAPT P10636 2/20 0.41
PTGS2 P35354 2/20 0.41
KDM4E B2RXH2 1/20 0.41
THRB P10828 1/20 0.41
ALOX15 P16050 1/20 0.41
NFKB1 P19838 1/20 0.41
THPO P40225 1/20 0.41
RECQL P46063 1/20 0.41
BLM P54132 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GNPAT O15228 1/20 0.39
ACACB O00763 2/20 0.38
SLC22A6 Q4U2R8 1/20 0.38
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2766000 1.00 ALDH1A1 (0.45) ALDH1A1MTNR1AMTNR1BMAPTPTGS2
SCHEMBL4378947 1.00 ALDH1A1 (0.45) ALDH1A1MTNR1AMTNR1BMAPTPTGS2
SCHEMBL1668685 0.82 ALDH1A1 (0.50) ALDH1A1MTNR1AMTNR1BMAPTPTGS2
SCHEMBL6249964 0.82 SLC22A6 (0.39) ALDH1A1MAPTPTGS2SMN1; SMN2SLC22A6
SCHEMBL20230310 0.82 GNPAT (0.56) ALDH1A1MAPTPTGS2KDM4ETHRB
SCHEMBL18395913 0.81 MTNR1A (0.46) ALDH1A1MTNR1AMTNR1BMAPTPTGS2
SCHEMBL18394981 0.81 MTNR1A (0.46) ALDH1A1MTNR1AMTNR1BMAPTPTGS2
SCHEMBL18394986 0.81 MTNR1A (0.46) ALDH1A1MTNR1AMTNR1BMAPTPTGS2
SCHEMBL18395917 0.81 MTNR1A (0.46) ALDH1A1MTNR1AMTNR1BMAPTPTGS2
SCHEMBL10055894 0.78 ITGB3 (0.43) ALDH1A1MAPTPTGS2SLC22A6ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1639994-A2 Topical composition comprising N-acetylaldosamines or N-acetylamino acids Yu, Ruey J., Dr. (US) 2006-03-29 EP claimed
CN-112300017-B Racemization preparation method of chiral beta-amino acid and derivative thereof 浙江九洲药业股份有限公司 2023-06-09 CN disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
WO-2021062246-A1 CRF RECEPTOR ANTAGONISTS AND METHODS OF USE NEUROCRINE BIOSCIENCES, INC. (US) 2021-04-01 WO disclosed
CN-112300017-A Racemization preparation method of chiral beta-amino acid and derivative thereof 浙江九洲药业股份有限公司 2021-02-02 CN disclosed
US-10252997-B2 Monocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-04-09 US disclosed
US-20180079723-A1 MONOCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-22 US disclosed
EP-3279183-A1 MONOCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2018-02-07 EP disclosed
US-9271993-B2 Treatment of bacterial infectious diseases UNIVERSITY OF ZURICH (CH) 2016-03-01 US disclosed
EP-2616079-B1 TREATMENT OF BACTERIAL INFECTIOUS DISEASES UNIV ZÜRICH (CH) 2015-10-14 EP disclosed
CN-1620294-A Pyrimidine A2BSelective antagonist compounds, their synthesis and use OSI PHARM INC (US) 2005-05-25 CN disclosed
US-20040186314-A1 Process for the preparation of enantiomerically enriched n-acyl-beta-amino acid derivatives by enantioselective hydrogenation of the corresponding (z)-enamides MALAN CHRISTOPHE GUILLAUME (CH) 2004-09-23 US disclosed
EP-1421059-A1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY ENRICHED N-ACYL-BETA-AMINO ACID DERIVATIVES BY ENANTIOSELECTIVE HYDROGENATION OF THE CORRESPONDING (Z)-ENAMIDES DOW GLOBAL TECHNOLOGIES INC. (US) 2004-05-26 EP disclosed
EP-1386901-A1 Method for producing an optically active beta-amino acid Takasago International Corporation (JP) 2004-02-04 EP disclosed
WO-2003016264-A1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY ENRICHED N-ACYL-BETA-AMINO ACID DERIVATIVES BY ENANTIOSELECTIVE HYDROGENATION OF THE CORRESPONDING (Z)-ENAMIDES CHIROTECH TECHNOLOGY LIMITED (GB) 2003-02-27 WO disclosed
US-6399787-B1 TRANSITION METAL COMPLEX PENN STATE RESEARCH FOUNDATION 2002-06-04 US disclosed
WO-1999059721-A1 CATALYTIC ASYMMETRIC HYDROGENATION, HYDROFORMYLATION, AND HYDROVINYLATION VIA TRANSITION METAL CATALYSTS WITH PHOSPHINES AND PHOSPHITES THE PENN STATE RESEARCH FOUNDATION (US) 1999-11-25 WO disclosed
US-5518903-A HYDROLYSIS OF ESTER CHISSO CORPORATION (JP) 1996-05-21 US disclosed
EP-0695296-A1 3-(HETERO)ARYLOXY(THIO) CARBOXYLIC ACID DERIVATIVES, METHOD OF PREPARING THEM AND INTERMEDIATES USED IN THEIR PREPARATION BASF AKTIENGESELLSCHAFT (DE) 1996-02-07 EP disclosed
WO-1994025443-A1 3-(HETERO)ARYLOXY(THIO) CARBOXYLIC ACID DERIVATIVES, METHOD OF PREPARING THEM AND INTERMEDIATES USED IN THEIR PREPARATION BASF AKTIENGESELLSCHAFT (DE) 1994-11-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10252997-B2 Monocyclic compound FABP1, CPT1A, GOT2 ALDH1A1 283/4885MTNR1A 995/4885MTNR1B 750/4885
US-20180079723-A1 MONOCYCLIC COMPOUND FABP1, CPT1A, GOT2 ALDH1A1 283/4885MTNR1A 995/4885MTNR1B 750/4885
US-20040186314-A1 Process for the preparation of enantiomerically enriched n-acyl-beta-amino acid derivatives by enantioselective hydrogenation of the corresponding (z)-enamides EEF1D, ADH5, HRH3 ALDH1A1 1084/4885MTNR1A 2147/4885MTNR1B 2480/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.