SCHEMBL7953606

SCHEMBL7953606

CN1CCN(c2cccc3[nH]c(C(=O)OCc4ccc(Cl)cc4)cc23)CC1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 1/20 0.50
MMP2 P08253 2/20 0.47
MMP1 P03956 1/20 0.47
MMP9 P14780 1/20 0.47
MMP12 P39900 1/20 0.47
HRH4 Q9H3N8 10/20 0.47
NPBWR1 P48145 1/20 0.44
MCHR1 Q99705 1/20 0.44
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
GAA P10253 2/20 0.40
MAPT P10636 1/20 0.40
RECQL P46063 1/20 0.40
ALOX5 P09917 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8818586 0.91 TMEM97 (0.50) MMP2MMP1MMP9MMP12HRH4
SCHEMBL7953556 0.89 TMEM97 (0.45) MMP2MMP1MMP9MMP12HRH4
SCHEMBL7943407 0.89 MMP9 (0.50) MMP2MMP1MMP9MMP12HRH4
SCHEMBL7949893 0.87 MMP12 (0.50) MMP1MMP12HRH4TMEM97SIGMAR1
SCHEMBL7949983 0.87 HTR1A (0.43) HRH4TMEM97SIGMAR1GAAMAPT
SCHEMBL7943428 0.87 MAPK1 (0.52) TMEM97SIGMAR1GAAMAPTALDH1A1
SCHEMBL7951610 0.86 HTR1A (0.44) GAAMAPTALDH1A1TSHR
SCHEMBL7943312 0.84 HRH4 (0.48) HRH4GAAMAPTALDH1A1
SCHEMBL7951589 0.82 KMT2A (0.51) OPRL1HRH4NPBWR1MCHR1MAPT
SCHEMBL7953632 0.81 HRH4 (0.54) HRH4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6255306-B1 PSYCHOLOGICAL DISORDERS MACOR JOHN E (US) 2001-07-03 US claimed
US-6255306-B1 PSYCHOLOGICAL DISORDERS MACOR JOHN E (US) 2001-07-03 US disclosed
EP-0773942-A1 4-INDOLE DERIVATIVES AS SEROTONIN AGONISTS AND ANTAGONISTS PFIZER INC. (US) 1997-05-21 EP disclosed
WO-1996003400-A1 4-INDOLE DERIVATIVES AS SEROTONIN AGONISTS AND ANTAGONISTS PFIZER INC. (US) 1996-02-08 WO disclosed