SCHEMBL7954472

SCHEMBL7954472

CC(C)Oc1cccc(CC(=O)N2CCCC(c3ccc(Cl)c(Cl)c3)C2CCS(C)(=O)=O)c1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
UTS2R Q9UKP6 5/20 0.48
TACR1 P25103 2/20 0.44
OPRK1 P41145 5/20 0.42
TACR2 P21452 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8592265 0.83 UTS2R (0.50) UTS2RTACR1OPRK1TACR2CYP3A4
SCHEMBL8806880 0.81 TACR1 (0.44) TACR1TACR2
SCHEMBL7954954 0.80 OPRK1 (0.42) TACR1OPRK1CYP3A4CYP2D6
SCHEMBL8592264 0.77 TACR1 (0.44) UTS2RTACR1OPRK1TACR2
SCHEMBL29790470 0.76 PPARA (0.54) TACR1TACR2
SCHEMBL8302191 0.74 POLB (0.51)
SCHEMBL8885666 0.73 TACR1 (0.38) TACR1OPRK1TACR2
SCHEMBL8885672 0.73 TACR1 (0.38) TACR1OPRK1TACR2
SCHEMBL7956616 0.72 TACR2 (0.44) UTS2RTACR1TACR2CYP3A4
SCHEMBL8308100 0.70 TACR1 (0.61) TACR1TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329392-B1 ANTIALLERGENS AVENTIS PHARMACEUTICALS, INC. 2001-12-11 US disclosed
WO-1996006094-A1 NOVEL SUBSTITUTED PIPERIDINES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES MERRELL PHARMACEUTICALS INC. (US) 1996-02-29 WO disclosed