SCHEMBL7955068

SCHEMBL7955068

Ic1ccc2c(C3CCNCC3)nsc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 6/20 0.40
CYP1A2 P05177 3/20 0.40
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
KCNH2 Q12809 1/20 0.33
SLC18A3 Q16572 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
QDPR P09417 1/20 0.31
TLR9 Q9NR96 3/20 0.31
TLR8 Q9NR97 3/20 0.31
TLR7 Q9NYK1 3/20 0.31
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1545776 0.82 CYP1A2 (0.41) GRM4CYP1A2
Hydrochloric Acid SCHEMBL6221807 0.81 CYP1A2 (0.41) GRM4CYP1A2
SCHEMBL1545124 0.78 KDM4E (0.49) GRM4CYP1A2MEN1KMT2AHTR2A
Hydrochloric Acid SCHEMBL1838069 0.77 KDM4E (0.51) GRM4CYP1A2MEN1KMT2AHTR2A
SCHEMBL7963908 0.77 CRHBP (0.39) GRM4CYP1A2MEN1KMT2ANPC1
SCHEMBL7954724 0.73 MKNK1 (0.40) NPC1RAB9A
SCHEMBL7966100 0.71 MAPK14 (0.47) GRM4CYP1A2HTR2ADRD2
SCHEMBL7966944 0.70 TLR9 (0.36) NPC1RAB9AHTR2ATLR9TLR8
SCHEMBL7962541 0.69 MKNK1 (0.33)
SCHEMBL1941279 0.68 HSP90AB1 (0.44) GRM4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303627-B1 FOR THERAPY OF PHYSIOLOGICAL AND PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY 2001-10-16 US disclosed
EP-0965587-A1 Tetrahydropyridinyl- and piperidinyl Inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1999-12-22 EP disclosed