SCHEMBL7956436

SCHEMBL7956436

N#Cc1ccc(C(NC(N)=O)c2ccccc2N2CCN(c3ccncc3)CC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PANK3 Q9H999 1/20 0.39
ALDH1A1 P00352 2/20 0.39
HTR1A P08908 2/20 0.38
DRD2 P14416 2/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38
PRSS1 P07477 1/20 0.38
CCR5 P51681 1/20 0.37
HRH1 P35367 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
MMP1 P03956 1/20 0.37
PARP1 P09874 1/20 0.36
AOC3 Q16853 1/20 0.35
NAMPT P43490 2/20 0.35
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7947608 0.87 MEN1 (0.42) ALDH1A1HTR1ADRD2GAAF2
SCHEMBL6429959 0.71 LMNA (0.64) ALDH1A1GAAPRSS1
SCHEMBL7947310 0.70 MCOLN3 (0.50) GAAMMP1NAMPT
SCHEMBL7956560 0.69 KDM4E (0.65) PANK3POLBHRH1HRH3
SCHEMBL10677218 0.69 CNR2 (0.47) ALDH1A1HTR1ADRD2GAAMMP1
SCHEMBL7956445 0.68 NAMPT (0.52) PANK3HTR1ADRD2NAMPTROCK2
SCHEMBL10635190 0.68 CNR2 (0.44) HTR1ADRD2POLBGAAMMP1
SCHEMBL7956239 0.67 CYP19A1 (0.46) GAAHRH1HRH3NAMPT
SCHEMBL7954927 0.67 HRH1 (0.52) ALDH1A1HTR1AHRH1HRH3
SCHEMBL7947472 0.67 SMN1; SMN2 (0.43) ALDH1A1GAAF2F10PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313127-B1 FOR THERAPY OF HYPERCHOLESTEROLEMIA OR ATHEROSCLEROSIS ZENECA LIMITED (GB) 2001-11-06 US disclosed
EP-0880501-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1998-12-02 EP disclosed
WO-1997028128-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1997-08-07 WO disclosed