SCHEMBL7961401

SCHEMBL7961401

COc1c2c(c(OC)c(OC)c1OC)CC(CCCOc1ccc(C(=O)O)cc1)C2

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.49
TSHR P16473 1/20 0.49
PLA2G4B P0C869 6/20 0.48
PKM P14618 1/20 0.47
RARB P10826 4/20 0.46
HTT P42858 1/20 0.46
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
NPC1 O15118 1/20 0.45
POLB P06746 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PLA2G4A P47712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7974351 0.96 TP53 (0.51) TP53TSHRPLA2G4BPKMRARB
SCHEMBL7961494 0.89 MAPT (0.56) HTTL3MBTL1NPC1POLBRAB9A
SCHEMBL7971231 0.86 GPR119 (0.53) L3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL7972638 0.85 MAPT (0.55) HTTL3MBTL1NPC1RAB9ASMN1; SMN2
SCHEMBL7971192 0.83 GPR119 (0.57) L3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL7974717 0.82 PKM (0.48) TP53TSHRPLA2G4BPKMRARB
SCHEMBL7972769 0.82 MAPT (0.47) L3MBTL1ALDH1A1KMT2A
SCHEMBL7973158 0.81 MEN1 (0.46) TP53TSHRPLA2G4BPKMRARB
SCHEMBL7977465 0.79 TP53 (0.49) TP53TSHRPLA2G4BPKMRARB
SCHEMBL7971292 0.78 HRH3 (0.41) TP53L3MBTL1NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326369-B1 ALZHEIMER'S DISEASE TAKEDA CHEMICALS INDUSTRIES, LTD. (JP) 2001-12-04 US disclosed
EP-0968164-A1 BICYCLIC QUINONE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2000-01-05 EP disclosed
WO-1998033758-A1 BICYCLIC QUINONE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-06 WO disclosed