SCHEMBL7973158

SCHEMBL7973158

COc1c2c(c(OC)c(OC)c1OC)CCC(CCOc1ccc(C(=O)O)cc1)CC2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PKM P14618 1/20 0.46
MAPK1 P28482 2/20 0.45
TSHR P16473 2/20 0.45
TP53 P04637 1/20 0.45
PLA2G4B P0C869 3/20 0.44
NPC1 O15118 1/20 0.44
POLB P06746 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
RARB P10826 4/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
USP2 O75604 1/20 0.43
ALOX15 P16050 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTT P42858 1/20 0.42
ALDH1A1 P00352 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7974462 0.86 MAPT (0.47) KMT2ARAB9AALDH1A1L3MBTL1
SCHEMBL833819 0.82 PKM (0.61) MEN1KMT2APKMMAPK1TSHR
SCHEMBL7972868 0.82 HRH3 (0.41)
SCHEMBL7972863 0.82 HRH3 (0.46) MAPK1NPC1RAB9A
SCHEMBL7977073 0.82 SIGMAR1 (0.44)
SCHEMBL7961401 0.81 TP53 (0.49) MEN1KMT2APKMMAPK1TSHR
SCHEMBL7974477 0.81 PKM (0.47) MEN1KMT2APKMMAPK1TSHR
SCHEMBL7961099 0.80 TP53 (0.46) MEN1KMT2APKMTSHRTP53
SCHEMBL7974351 0.80 TP53 (0.51) MEN1KMT2APKMMAPK1TSHR
SCHEMBL7316232 0.78 NFE2L2 (0.62) MEN1KMT2APKMMAPK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326369-B1 ALZHEIMER'S DISEASE TAKEDA CHEMICALS INDUSTRIES, LTD. (JP) 2001-12-04 US disclosed
EP-0968164-A1 BICYCLIC QUINONE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2000-01-05 EP disclosed
WO-1998033758-A1 BICYCLIC QUINONE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-06 WO disclosed