SCHEMBL7962457

SCHEMBL7962457

COC(=O)[C@H](Cc1ccc2c(c1)oc1ccccc12)NC(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.53
ECE1 P42892 7/20 0.51
MME P08473 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
EPHX2 P34913 1/20 0.49
CTSS P25774 5/20 0.47
CTSK P43235 4/20 0.47
CTSB P07858 3/20 0.47
ACE P12821 1/20 0.46
CTSL P07711 1/20 0.45
TACR1 P25103 1/20 0.45
KDR P35968 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7962462 1.00 KLK5 (0.53) KLK5ECE1MMEMEN1KMT2A
SCHEMBL7962403 0.90 ECE1 (0.60) ECE1MMEMEN1KMT2ACTSS
SCHEMBL7972346 0.90 ECE1 (0.60) ECE1MMEMEN1KMT2ACTSS
SCHEMBL7972340 0.87 ECE1 (0.44) KLK5ECE1MMEMEN1KMT2A
SCHEMBL7972405 0.85 ECE1 (0.55) ECE1MMEMEN1KMT2ATACR1
SCHEMBL7975670 0.85 ECE1 (0.55) ECE1MMEMEN1KMT2ATACR1
SCHEMBL5630007 0.80 CTSS (0.69) KLK5MEN1KMT2ACTSSCTSK
SCHEMBL31584535 0.80 CTSS (0.69) KLK5MEN1KMT2ACTSSCTSK
SCHEMBL7976231 0.79 ECE1 (0.49) ECE1MMEMEN1KMT2AKDR
SCHEMBL5115337 0.79 CA12 (0.49) KLK5KMT2AEPHX2CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001077095-A2 DERIVATIVES OF ALPHA-MERCAPTOACETAMIDE NOVARTIS AG (CH) 2001-10-18 WO disclosed