SCHEMBL7963938

SCHEMBL7963938

Cn1nc(C(F)(F)F)cc1Oc1cccc(C(=O)NCC(F)(F)F)n1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
SCN9A Q15858 4/20 0.41
SCN10A Q9Y5Y9 2/20 0.41
MAPT P10636 1/20 0.40
P2RX7 Q99572 1/20 0.40
EGLN2 Q96KS0 1/20 0.39
KMT2A Q03164 1/20 0.39
DDR1 Q08345 1/20 0.39
IRAK4 Q9NWZ3 6/20 0.38
ULK1 O75385 1/20 0.37
FLT3 P36888 1/20 0.37
CYP3A4 P08684 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TGFBR1 P36897 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8720573 0.85 KMT2A (0.39) ALDH1A1ADORA2AADORA1SCN9ASCN10A
SCHEMBL8574398 0.83 ADORA2A (0.50) ALDH1A1ADORA2AADORA1MAPTKMT2A
SCHEMBL7964413 0.82 MAPT (0.50) ALDH1A1ADORA2AADORA1MAPTKMT2A
SCHEMBL5553184 0.75 ADORA2A (0.49) ALDH1A1ADORA2AADORA1KMT2ATGFBR1
SCHEMBL6615519 0.74 ALDH1A1 (0.40) ALDH1A1ADORA2AADORA1EGLN2KMT2A
SCHEMBL7953446 0.74 KMT2A (0.50) ALDH1A1ADORA2AADORA1MAPTKMT2A
SCHEMBL6613473 0.73 ADORA2A (0.44) ALDH1A1ADORA2AADORA1KMT2ATGFBR1
SCHEMBL6613296 0.73 ADORA2A (0.48) ALDH1A1ADORA2AADORA1KMT2ATGFBR1
SCHEMBL9017235 0.73 SCN9A (0.46) SCN9ASCN10AKMT2AULK1
SCHEMBL6614783 0.72 ADORA2A (0.41) ALDH1A1ADORA2AADORA1MAPTEGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7285962-A None JP disclosed
US-6271372-B1 REACTING HETEROAROMATIC HALOGEN COMPOUNDS WITH CARBON MONOXIDE AND AROMATIC AMINES IN THE PRESENCE OF A COMPLEX OF PALLADIUM WITH A TRIPHENYLPHOSPHINE AND A BASE OTHER THAN AN AMINE. LONZA AG (CH) 2001-08-07 US disclosed
US-5900484-A FROM HETEROAROMATIC HALOGEN COMPOUNDS AND AROMATIC AMINES AND CARBON MONOXIDE WITH PALLADIUM PHOSPHINE COMPLEX LONZA AG (CH) 1999-05-04 US disclosed
JP-H07285962-A PYRIDINECARBOXYLIC ACID AMIDE DERIVATIVE NISSAN CHEM IND LTD 1995-10-31 JP disclosed