SCHEMBL7963943

SCHEMBL7963943

Cc1ccc(N2CCN(CCCc3nn(-c4ccccc4)c4c3CCCC4)CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
SIGMAR1 Q99720 4/20 0.47
KCNH2 Q12809 3/20 0.46
HTR7 P34969 1/20 0.44
HTR1A P08908 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963930 0.93 SIGMAR1 (0.53) SIGMAR1KCNH2HTR7HTR1APTGS1
SCHEMBL7959679 0.89 DRD3 (0.49) SIGMAR1KCNH2HTR7HTR1A
SCHEMBL7957403 0.85 MAPT (0.46) MAPTNPSR1SIGMAR1KCNH2HTR7
SCHEMBL7959137 0.84 SIGMAR1 (0.53) SIGMAR1KCNH2HTR7HTR1A
Fumaric Acid SCHEMBL7959573 0.83 SIGMAR1 (0.49) SIGMAR1HTR7HTR1APTGS1PTGS2
Maleic Acid SCHEMBL7959572 0.83 SIGMAR1 (0.49) SIGMAR1HTR7HTR1APTGS1PTGS2
SCHEMBL15961278 0.76 SIGMAR1 (0.79) MAPTNPSR1SIGMAR1KCNH2HTR7
SCHEMBL7959536 0.76 SIGMAR1 (0.52) SIGMAR1HTR7HTR1A
SCHEMBL7959986 0.76 HTR1A (0.51) SIGMAR1HTR1ASLC6A3
SCHEMBL7963946 0.74 MAPT (0.46) MAPTNPSR1SIGMAR1KCNH2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187774-B1 N-PIPERAZINYLALKYLINDAZOLE DERIVATIVES; PSYCHOLOGICAL DISORDERS, SCHIZOPHRENIA; SIDE EFFECT REDUCTION YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2001-02-13 US disclosed
EP-0885883-A1 FUSED HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL APPLICATIONS THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1998-12-23 EP disclosed