SCHEMBL7963930

SCHEMBL7963930

c1ccc(N2CCN(CCCc3nn(-c4ccccc4)c4c3CCCC4)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.53
KCNH2 Q12809 2/20 0.51
PTGS2 P35354 3/20 0.48
PTGS1 P23219 2/20 0.48
CYP2D6 P10635 1/20 0.48
DRD2 P14416 4/20 0.46
HTR1A P08908 2/20 0.46
DRD3 P35462 2/20 0.46
DRD4 P21917 1/20 0.46
HTR2A P28223 1/20 0.45
HRH1 P35367 1/20 0.45
TMEM97 Q5BJF2 1/20 0.45
HTR7 P34969 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963943 0.93 MAPT (0.50) SIGMAR1KCNH2PTGS2PTGS1HTR1A
SCHEMBL7959679 0.93 DRD3 (0.49) SIGMAR1KCNH2DRD2HTR1ADRD3
SCHEMBL7959137 0.88 SIGMAR1 (0.53) SIGMAR1KCNH2CYP2D6DRD2HTR1A
Fumaric Acid SCHEMBL7959573 0.86 SIGMAR1 (0.49) SIGMAR1PTGS2PTGS1DRD2HTR1A
Maleic Acid SCHEMBL7959572 0.86 SIGMAR1 (0.49) SIGMAR1PTGS2PTGS1DRD2HTR1A
SCHEMBL7957403 0.77 MAPT (0.46) SIGMAR1KCNH2DRD2HTR1ADRD3
SCHEMBL7959986 0.76 HTR1A (0.51) SIGMAR1DRD2HTR1ADRD3DRD4
SCHEMBL7959536 0.76 SIGMAR1 (0.52) SIGMAR1DRD2HTR1ADRD3DRD4
SCHEMBL10479713 0.76 PTGS2 (0.51) PTGS2PTGS1CYP2D6
SCHEMBL10479760 0.76 PTGS2 (0.60) PTGS2PTGS1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187774-B1 N-PIPERAZINYLALKYLINDAZOLE DERIVATIVES; PSYCHOLOGICAL DISORDERS, SCHIZOPHRENIA; SIDE EFFECT REDUCTION YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2001-02-13 US disclosed
EP-0885883-A1 FUSED HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL APPLICATIONS THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1998-12-23 EP disclosed