SCHEMBL7965741

SCHEMBL7965741

O[C@H](COc1cccc2[nH]ccc12)CN1CCC(O)(c2cncc3ccccc23)CC1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 18/20 0.54
SLC6A4 P31645 4/20 0.54
ADRB2 P07550 1/20 0.51
ADRB1 P08588 1/20 0.51
ADRB3 P13945 1/20 0.51
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7814249 0.90 HTR1A (0.58) HTR1ASLC6A4ADRB2ADRB1ADRB3
SCHEMBL7962445 0.85 HTR1A (0.42) HTR1ASLC6A4
SCHEMBL7965744 0.83 HTR1A (0.36) HTR1ASLC6A4ADRB2ADRB1ADRB3
SCHEMBL7965737 0.83 HTR1A (0.41) HTR1ASLC6A4ADRB2ADRB1
SCHEMBL7953370 0.83 HTR1A (0.56) HTR1ASLC6A4ADRB2ADRB1ADRB3
SCHEMBL7887623 0.82 ABCB1 (0.61) HTR1ASLC6A4ADRB2ADRB1ADRB3
SCHEMBL5584644 0.82 HTR1A (0.59) HTR1ASLC6A4ADRB2ADRB1ADRB3
SCHEMBL7964959 0.82 HTR1A (0.69) HTR1ASLC6A4ADRB2ADRB1ADRB3
SCHEMBL7953974 0.81 HTR1A (0.41) HTR1ASLC6A4ADRB1CYP1A2CYP2C19
SCHEMBL7965451 0.79 SMN1; SMN2 (0.55) HTR1ACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed
EP-0976747-A2 Use of 5HT-1F receptor antagonists for treating anxiety disorders ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed