SCHEMBL7966843

SCHEMBL7966843

c1ccc(CN2CCN(c3ccccc3-c3nc(-c4ccccc4)no3)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.63
KCNH2 Q12809 1/20 0.63
ALDH1A1 P00352 5/20 0.58
CASP1 P29466 1/20 0.58
CASP7 P55210 1/20 0.58
LMNA P02545 5/20 0.54
MAPT P10636 5/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
TSHR P16473 1/20 0.54
HSD17B10 Q99714 1/20 0.54
S1PR1 P21453 2/20 0.50
GPR55 Q9Y2T6 1/20 0.50
ACHE P22303 1/20 0.50
S1PR4 O95977 1/20 0.50
S1PR5 Q9H228 1/20 0.50
DRD2 P14416 3/20 0.49
HTR1A P08908 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
TDP1 Q9NUW8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7961623 0.82 MAPT (0.62) ALDH1A1CASP1CASP7LMNAMAPT
SCHEMBL17100583 0.81 CYP2D6 (0.71) CYP2D6KCNH2ALDH1A1CASP1CASP7
SCHEMBL5734895 0.80 HTR7 (0.61) ALDH1A1LMNAMAPTSMN1; SMN2TSHR
SCHEMBL7821576 0.75 MAPT (0.50) ALDH1A1MAPTTSHRDRD2HTR1A
SCHEMBL23958379 0.74 CYP2D6 (0.92) CYP2D6KCNH2ALDH1A1CASP1CASP7
SCHEMBL17100616 0.73 LMNA (0.67) CYP2D6KCNH2ALDH1A1CASP1CASP7
SCHEMBL5736286 0.72 MAPT (0.53) ALDH1A1MAPTSMN1; SMN2S1PR1GPR55
SCHEMBL8611543 0.72 DRD4 (0.60) CYP2D6KCNH2ALDH1A1LMNAMAPT
SCHEMBL17100611 0.71 MAPK1 (0.57) CYP2D6KCNH2ALDH1A1CASP1CASP7
SCHEMBL17100655 0.71 MAPT (0.66) CYP2D6KCNH2ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6277872-B1 ANTIISCHEMIC AGENTS; BRAIN DISORDERS BOEHRINGER INGELHEIM KG (DE) 2001-08-21 US disclosed