SCHEMBL7973908

SCHEMBL7973908

CCOC(=O)c1csc(-c2ccc(C(c3cccc(O)c3)N3CCN4CCC[C@@H]4C3)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.41
GAA P10253 1/20 0.41
CLK1 P49759 2/20 0.40
NPC1 O15118 2/20 0.40
KMT2A Q03164 4/20 0.38
KDM4E B2RXH2 2/20 0.38
RXFP1 Q9HBX9 2/20 0.38
OGA O60502 1/20 0.38
MEN1 O00255 3/20 0.37
POLB P06746 3/20 0.37
ALDH1A1 P00352 2/20 0.37
OPRD1 P41143 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36
SLC6A9 P48067 3/20 0.36
PIN1 Q13526 1/20 0.36
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7967499 0.88 RAB9A (0.40) RAB9AGAACLK1NPC1KMT2A
SCHEMBL7968969 0.83 KDM4E (0.41) GAAKMT2AKDM4EMEN1POLB
SCHEMBL7957883 0.78 RAB9A (0.43) RAB9AGAACLK1NPC1RXFP1
SCHEMBL7970812 0.77 CYP1A2 (0.48) RAB9AGAAOPRD1CYP3A4
SCHEMBL7968609 0.77 PIN1 (0.41) ALDH1A1OPRD1CYP3A4PIN1HPGDS
SCHEMBL7967851 0.76 CYP1A2 (0.45) OPRD1CYP3A4
SCHEMBL7968921 0.75 OPRD1 (0.60) OPRD1CYP3A4
SCHEMBL7968646 0.69 OPRD1 (0.51) OPRD1
SCHEMBL28154886 0.69 RAB9A (0.70) RAB9AGAACLK1NPC1KMT2A
SCHEMBL29911269 0.68 RAB9A (0.66) RAB9AGAACLK1NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6200978-B1 FOR PREVENTING OR TREATING INFLAMMATORY DISEASES SUCH AS ARTHRITIS, PSORIASIS, ASTHMA, OR INFLAMMATORY BOWEL DISEASE, DISORDERS OF RESPIRATORY FUNCTION, GASTROINTESTINAL DISORDERS SUCH AS FUNCTIONAL BOWEL DISEASE, AS ANALGESICS PFIZER INC. 2001-03-13 US disclosed